Exenatide (Byetta)

Category: GLP-1 Agonist

First-in-class GLP-1 receptor agonist derived from Gila monster venom, used for type 2 diabetes.

Half-Life: 2.4 hours

Benefits

  • Blood sugar control
  • Modest weight loss
  • Twice daily or weekly formulations available
  • Cardiovascular benefits

Side Effects

  • Nausea
  • Vomiting
  • Diarrhea
  • Injection site reactions
  • Pancreatitis risk